《分子药理学杂志》.2005年.第5期

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• Concurrent Stimulation of Cannabinoid CB1 and Dopamine D2 Receptors Enhances Heterodimer Formation: A Mechanism for Receptor Cross-Talk
• 2-Adrenergic Agonist Enrichment of Spinophilin at the Cell Surface Involves Subunits of Gi Proteins and Is Preferentially Induced by the 2A
• Polyspecific Organic Cation Transport: Insights into the Substrate Binding Site
• The Met852 Residue Is a Key Organizer of the Ligand-Binding Cavity of the Human Mineralocorticoid Receptor
• Subtype-Specific Sorting of the ETA Endothelin Receptor by a Novel Endocytic Recycling Signal for G Protein-Coupled Receptors
• A Novel and Efficient Approach to Discriminate between Pre- and Post-Transcription HIV Inhibitors
• Superagonistic Action of 14-epi-Analogs of 1,25-Dihydroxyvitamin D Explained by Vitamin D Receptor-Coactivator Interaction
• The Human Organic Anion Transporter 2 Gene Is Transactivated by Hepatocyte Nuclear Factor-4 and Suppressed by Bile Acids
• Subtype-Specific Affinity for Corticosterone of Rat Organic Cation Transporters rOCT1 and rOCT2 Depends on Three Amino Acids within the Subs
• The General Anesthetic Isoflurane Depresses Synaptic Vesicle Exocytosis
• Internal PDZ Ligands: Novel Endocytic Recycling Motifs for G Protein-Coupled Receptors
• Pharmacological Discrimination of Calcitonin Receptor: Receptor Activity-Modifying Protein Complexes
• Differential Modulation of Glutamatergic Transmission by 3,5-Dibromo-L-phenylalanine
• Long-Term Nicotine Treatment Decreases Striatal 6 Nicotinic Acetylcholine Receptor Sites and Function in Mice
• Transcriptional Regulation of Mouse eOpioid Receptor Gene: Sp3 Isoforms(M1, M2) Function as Repressors in Neuronal Cells to Regulate the eO
• Amino Acids Critical for Substrate Affinity of Rat Organic Cation Transporter 1 Line the Substrate Binding Region in a Model Derived from th
• Effect of Azelnidipine on Angiotensin II-Mediated Growth-Promoting Signaling in Vascular Smooth Muscle Cells
• Potentiation of P2Y Receptors by Physiological Elevations of Extracellular K+ via a Mechanism Independent of Ca2+ Influx
• Constitutive Activation and Environmental Chemical Induction of the Aryl Hydrocarbon Receptor/Transcription Factor in Activated Human B Lymp
• Identification and Characterization of a Functional TATA Box Polymorphism of the UDP Glucuronosyltransferase 1A7 Gene
• The Breast Cancer Resistance Protein(BCRP/ABCG2) Affects Pharmacokinetics, Hepatobiliary Excretion, and Milk Secretion of the Antibiotic Ni
• The Aminosteroid Phospholipase C Antagonist U-73122(1-[6-[[17--3-Methoxyestra-1,3,5(10)-trien-17-yl]amino]hexyl]-1H-pyrrole-2,5-dione) Pote
• A Natural CYP2B6 TATA Box Polymorphism(eC82T C) Leading to Enhanced Transcription and Relocation of the Transcriptional Start Site
• Sex-Dependent Expression and Activity of the ATP-Binding Cassette Transporter Breast Cancer Resistance Protein(BCRP/ABCG2) in Liver
• Phenylglycine and Sulfonamide Correctors of Defective F508 and G551D Cystic Fibrosis Transmembrane Conductance Regulator Chloride-Channel Ga
• Developmental Regulation of -Carboline-Induced Inhibition of Glycine-Evoked Responses Depends on Glycine Receptor Subunit Expression
• Aspects of Dioxin Toxicity Are Mediated by Interleukin 1-Like Cytokines
• The Effect of Hydroxylamine on KATP Channels in Vascular Smooth Muscle and Underlying Mechanisms
• Expression of the Retinoic Acid-Metabolizing Enzyme CYP26A1 Limits Programmed Cell Death
• Mechanism of the Anti-Inflammatory Effect of Thiazolidinediones: Relationship with the Glucocorticoid Pathway
• Cephalostatin 1 Inactivates Bcl-2 by Hyperphosphorylation Independent of M-Phase Arrest and DNA Damage
• Heparan Sulfate Regulates the Antiangiogenic Activity of Endothelial Monocyte-Activating Polypeptide-II at Acidic pH
• Adenosine A2A Receptor Stimulation Increases Angiogenesis by Down-Regulating Production of the Antiangiogenic Matrix Protein Thrombospondin
• U937 Cell Necrosis Mediated by Peroxynitrite Is Not Caused by Depletion of ATP and Is Prevented by Arachidonate via an ATP-Dependent Mechani
• The Repertoire of G-ProteineCCoupled Receptors in Fully Sequenced Genomes
• Adenosine in Tissue Protection and Tissue Regeneration
• Effects of Valproic Acid Derivatives on Inositol Trisphosphate Depletion, Teratogenicity, Glycogen Synthase Kinase-3 Inhibition, and Viral R
• Vacuolar Degradation of Rat Liver CYP2B1 in Saccharomyces cerevisiae: Further Validation of the Yeast Model and Structural Implications for
• Blockade of Vascular Endothelial Growth Factor Receptor Signal Pathway and Antitumor Activity of ON-III(2',4'-Dihydroxy-6'-methoxy-3',5'-di
• Palmitoylation of the 5-Hydroxytryptamine4a Receptor Regulates Receptor Phosphorylation, Desensitization, and -Arrestin-Mediated Endocytosis
• Modulation of Cellular Response to Cisplatin by a Novel Inhibitor of DNA Polymerase
• Structural Features of the Glutamate Binding Site in Recombinant NR1/NR2A N-Methyl-D-aspartate Receptors Determined by Site-Directed Mutagen
• Antiangiogenic and Vascular-Targeting Activity of the Microtubule-Destabilizing trans-Resveratrol Derivative 3,5,4'-Trimethoxystilbene
• Investigations of Calsequestrin as a Target for Anthracyclines: Comparison of Functional Effects of Daunorubicin, Daunorubicinol, and Triflu
• -Adrenergic Receptor Stimulation Promotes Gs Internalization through Lipid Rafts: A Study in Living Cells
• From Plants to Man: The GPCR "Tree of Life"
• Isoflurane Induces a Protein Kinase C -Dependent Increase in Cell-Surface Protein Level and Activity of Glutamate Transporter Type 3
• Stichodactyla helianthus Peptide, a Pharmacological Tool for Studying Kv3.2 Channels
• Marked Depletion of Glycosylation Sites in HIV-1 gp120 under Selection Pressure by the Mannose-Specific Plant Lectins of Hippeastrum Hybrid
• A Synthetic Derivative of the Natural Product Rocaglaol Is a Potent Inhibitor of Cytokine-Mediated Signaling and Shows Neuroprotective Activ